(-)-Sparteine sulfate pentahydrate ( —— )

产品货号. M15325 CAS No. 6160-12-9

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

(-)-Sparteine sulfate pentahydrate
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

金雀花碱是 1a 类抗心律失常药；钠通道阻滞剂。它是一种生物碱，可以从金雀花中提取。
产品描述

Sparteine is a class 1a antiarrhythmic agent; a sodium channel blocker. It is an alkaloid and can be extracted from scotch broom. It is the predominant alkaloid in Lupinus mutabilis, and is thought to chelate the bivalents calcium and magnesium. It is not FDA approved for human use as an antiarrhythmic agent, and it is not included in the Vaughn Williams classification of antiarrhythmic drugs.
体外实验

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体内实验

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同义词

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通路

Metabolic Enzyme/Protease
靶点

P450
受体

CYP2D
研究领域

Cardiovascular Disease
适应症

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1.Preissner S, et al. Nucleic Acids Res. 2010 Jan; 38(Database issue):D237-43.

计算器

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